Synthesis and Biological Evaluation of N-((1-(4-(Sulfonyl)piperazin-1-yl)cycloalkyl)methyl)benzamide Inhibitors of Glycine Transporter-1

Cioffi, Christopher L.; Liu, Shuang; Wolf, Mark A.; Guzzo, Peter R.; Sadalapure, Kashinath; Parthasarathy, Visweswaran; Loong, David T.J.; Maeng, Jun-Ho; Carulli, Edmund; Fang, Xiao; Karunakaran, Kalesh; Matta, Lakshman; Choo, Sok Hui; Panduga, Shailijia; Buckle, Ronald N.; Davis, Randall N.; Sakwa, Samuel A.; Gupta, Priya; Sargent, Bruce J.; Moore, Nicholas A.; Luche, Michele M.; Carr, Grant J.; Khmelnitsky, Yuri L.; Ismail, Jiffry; Chung, Mark; Bai, Mei; Leong, Wei Yee; Sachdev, Nidhi; Swaminathan, Srividya; Mhyre, Andrew J.

doi:10.1021/acs.jmedchem.6b00914

All Outputs (3)

A capillary electrophoresis method to explore the self-assembly of a novel polypeptide ligand with quantum dots (2016)
Journal Article
Wang, J., Zhang, C., Liu, L., Kalesh, K. A., Qiu, L., Ding, S., …Jiang, P. (2016). A capillary electrophoresis method to explore the self-assembly of a novel polypeptide ligand with quantum dots. ELECTROPHORESIS, 37(15-16), https://doi.org/10.1002/elps.201600164

Target identification of natural and traditional medicines with quantitative chemical proteomics approaches (2016)
Journal Article
Wang, J., Gao, L., Lee, Y. M., Kalesh, K. A., Ong, Y. S., Lim, J., …Lin, Q. (2016). Target identification of natural and traditional medicines with quantitative chemical proteomics approaches. Pharmacology and Therapeutics, 162, https://doi.org/10.1016/j.pharmthera.2016.01.010

Synthesis and Biological Evaluation of N-((1-(4-(Sulfonyl)piperazin-1-yl)cycloalkyl)methyl)benzamide Inhibitors of Glycine Transporter-1 (2016)
Journal Article
Cioffi, C. L., Liu, S., Wolf, M. A., Guzzo, P. R., Sadalapure, K., Parthasarathy, V., …Mhyre, A. J. (2016). Synthesis and Biological Evaluation of N-((1-(4-(Sulfonyl)piperazin-1-yl)cycloalkyl)methyl)benzamide Inhibitors of Glycine Transporter-1. Journal of Medicinal Chemistry, 59(18), 8473-8494. https://doi.org/10.1021/acs.jmedchem.6b00914