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Functionalized pyridylboronic acids and their Suzuki cross-coupling reactions to yield novel heteroarylpyridines

Parry, P.R.; Wang, C.S.; Batsanov, A.S.; Bryce, M.R.; Tarbit, B.

Authors

P.R. Parry

C.S. Wang

A.S. Batsanov

B. Tarbit



Abstract

2-Bromo-5-pyridylboronic acid 2a, 2-chloro-5-pyridylboronic acid 2b, 2-methoxy-5-pyridylboronic acid 2c, and 5-chloro-2-methoxy-4-pyridylboronic acid 4 have been synthesized and shown to undergo palladium-catalyzed cross-coupling reactions with heteroaryl bromides to yield novel heteroarylpyridine derivatives. The X-ray crystal structures of 2a and 2b have been obtained.

Citation

Parry, P., Wang, C., Batsanov, A., Bryce, M., & Tarbit, B. (2002). Functionalized pyridylboronic acids and their Suzuki cross-coupling reactions to yield novel heteroarylpyridines. Journal of Organic Chemistry, 67(21), 7541-7543

Journal Article Type Article
Publication Date 2002-10
Journal Journal of Organic Chemistry
Print ISSN 0022-3263
Publisher American Chemical Society
Peer Reviewed Peer Reviewed
Volume 67
Issue 21
Pages 7541-7543