Giuliano Cesar Clososki
C-H activation/metalation approaches for the synthesis of indolizine derivatives
Clososki, Giuliano Cesar; Steel, Patrick G.; Bertallo, Camila Rodrigues de Souza; Arroio, Thaís Rodrigues Arroio Rodrigues; Vessecchi, Ricardo; Toledo, Monica F.Z.J.; Sadler, Scott
Authors
Professor Patrick Steel p.g.steel@durham.ac.uk
Professor
Camila Rodrigues de Souza Bertallo
Thaís Rodrigues Arroio Rodrigues Arroio
Ricardo Vessecchi
Monica F.Z.J. Toledo
Scott Sadler
Abstract
The C‐H borylation of indolizines has not previously been reported and in this communication, we describe our preliminary efforts to apply this chemistry to this scaffold and contrast this approach to directed metalation. Through these methodologies were possible obtain a library of substituted indolizines functionalized in both pyridinic and pyrrole ring.
Citation
Clososki, G. C., Steel, P. G., Bertallo, C. R. D. S., Arroio, T. R. A. R., Vessecchi, R., Toledo, M. F., & Sadler, S. (2019). C-H activation/metalation approaches for the synthesis of indolizine derivatives. European Journal of Organic Chemistry, 31-32, 5205-5213. https://doi.org/10.1002/ejoc.201900608
Journal Article Type | Article |
---|---|
Acceptance Date | Jun 5, 2019 |
Publication Date | Sep 30, 2019 |
Deposit Date | Jun 6, 2019 |
Publicly Available Date | Jun 25, 2020 |
Journal | European Journal of Organic Chemistry |
Print ISSN | 1434-193X |
Electronic ISSN | 1099-0690 |
Publisher | Wiley |
Peer Reviewed | Peer Reviewed |
Volume | 31-32 |
Pages | 5205-5213 |
DOI | https://doi.org/10.1002/ejoc.201900608 |
Public URL | https://durham-repository.worktribe.com/output/1300433 |
Files
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Copyright Statement
This is the accepted version of the following article: Clososki, Giuliano Cesar, Steel, Patrick G., Bertallo, Camila Rodrigues de Souza, Arroio, Thaís Rodrigues Arroio Rodrigues, Vessecchi, Ricardo, Toledo, Monica F. Z. J. & Sadler, Scott (2019). C-H activation/metalation approaches for the synthesis of indolizine derivatives. European Journal of Organic Chemistry 31-32: 5205-5213 which has been published in final form at https://doi.org/10.1002/ejoc.201900608. This article may be used for non-commercial purposes in accordance With Wiley Terms and Conditions for self-archiving.
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