Regioselective Functionalization of 7‐Azaindole by Controlled Annular Isomerism: The Directed Metalation‐Group Dance
(2019)
Journal Article
Snieckus, V., Patel, J., Kitching, M., Dalziel, M., Cosman, J., & Kaye, M. (2019). Regioselective Functionalization of 7‐Azaindole by Controlled Annular Isomerism: The Directed Metalation‐Group Dance. Angewandte Chemie, 131(22), 7391-7395. https://doi.org/10.1002/ange.201901724
The regioselective functionalization of 7‐azaindole by controlled annular directed metalation group isomerism is reported. The N‐7 carbamoyl azaindoles 2a–b undergo regioselective metalation and electrophile quench to furnish C‐6 substituted derivati... Read More about Regioselective Functionalization of 7‐Azaindole by Controlled Annular Isomerism: The Directed Metalation‐Group Dance.